Dihydropyrimidone Derivatives as Thymidine Phosphorylase Inhibitors: Inhibition Kinetics, Cytotoxicity, and Molecular Docking

Cui, TM; Altaf, M; Aldarhami, A; Bazaid, AS; Saeedi, NH; Alkayyal, AA; Alshabrmi, FM; Ali, F; Aladhadh, M; Khan, MY; Alsaiari, AA; Ma, YR

Ma, YR (通讯作者),Chengdu Univ Tradit Chinese Med, Sch Basic Med, Chengdu 610075, Peoples R China.;Aldarhami, A (通讯作者),Umm Al Qura Univ, Qunfudah Fac Med, Dept Med Microbiol, Al Qunfudah 21961, Saudi Arabia.

MOLECULES, 2023; 28 (8):

Abstract

Overexpression of the thymidine phosphorylase (TP) enzyme induces angiogenesis, which eventually leads to metastasis and tumor growth. The crucial rol......

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