Optimization of 4-amino-pyridazin-3(2H)-one as a valid core scaffold for FABP4 inhibitors

Floresta, G; Crocetti, L; Silva, RRD; Patamia, V; Mazzacuva, F; Chen, YCS; Vergelli, C; Cilibrizzi, A

Crocetti, L (通讯作者),Dept Neurofarba, Via Ugo Schiff 6, I-50019 Florence, Italy.;Cilibrizzi, A (通讯作者),Kings Coll London, Inst Pharmaceut Sci, Stamford St, London SE1 9NH, England.

ARCHIV DER PHARMAZIE, 2023; 356 (10):

Abstract

Current clinical research suggests that fatty acid-binding protein 4 inhibitors (FABP4is), which are of biological and therapeutic interest, may show ......

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