Comparative evaluation of biased agonists Sarcosine1, d-Alanine8-Angiotensin (Ang) II (SD Ang II) and Sarcosine1, Isoleucine8-Ang II (SI Ang II) and their radioiodinated congeners binding to rat liver membrane AT1 receptors

Noto, NM; Restrepo, YM; Pang, HW; Stoyell-Conti, F; West, CA; Speth, RC

West, CA (通讯作者),Appalachian State Univ, Dept Biol, North Carolina Res Campus,150 N Res Campus Dr Kann, Kannapolis, NC 28081 USA.;Speth, RC (通讯作者),Nova Southeastern Univ, Coll Pharm, 3200 S Univ Dr, Ft Lauderdale, FL 33328 USA.

PHARMACOLOGY RESEARCH & PERSPECTIVES, 2023; 11 (1):

Abstract

Angiotensin II analogue and beta-arrestin biased agonist TRV027 (Sarcosine(1), d-Alanine(8)-Angiotensin (Ang) II; SD Ang II), developed by Trevena, In......

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