Discovery of alkyl bis(oxy)dibenzimidamide derivatives as novel protein arginine methyltransferase 1 (PRMT1) inhibitors

Zhang, WY; Lu, WC; Jiang, H; Lv, ZB; Xie, YQ; Lian, FL; Liang, ZJ; Jiang, YX; Wang, DJ; Luo, C; Jin, J; Ye, F

Jin, J; Ye, F (reprint author), Zhejiang Sci Tech Univ, Coll Life Sci, Hangzhou, Zhejiang, Peoples R China.

CHEMICAL BIOLOGY & DRUG DESIGN, 2017; 90 (6): 1260

Abstract

Protein arginine methylation, a post-translational modification critical for a variety of biological processes, is catalyzed by protein arginine N-met......

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