Design, synthesis and anticancer activity studies of novel indole derivatives as Bcl-2/Mcl-1 dual inhibitors

Liu, YF; Li, JJ; Zhou, GH; Zhang, JL; Teng, Y; Bai, ZS; Liu, TT

Liu, TT (通讯作者),Shandong First Med Univ & Shandong Acad Med Sci, Sch Pharm, Dept Med Chem, Tai An 271016, Shandong, Peoples R China.;Bai, ZS (通讯作者),Shandong First Med Univ & Shandong Acad Med Sci, Inst Mat Med, Jinan 250000, Shandong, Peoples R China.

MEDICINAL CHEMISTRY RESEARCH, 2023; 32 (1): 99

Abstract

A series of novel indole derivatives were designed, synthesized and evaluated for the binding affinity of Bcl-2 family proteins and antiproliferative ......

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