Development of the First Covalent Monopolar Spindle Kinase 1 (MPS1/TTK) Inhibitor
Serafim, RAM; Santiago, AD; Schwalm, MP; Hu, ZX; dos Reis, CV; Takarada, JE; Mezzomo, P; Massirer, KB; Kudolo, M; Gerstenecker, S; Chaikuad, A; Zender, L; Knapp, S; Laufer, S; Counago, RM; Gehringer, M
Gehringer, M (通讯作者),Eberhard Karls Univ Tubingen, Dept Pharmaceut Med Chem, D-72076 Tubingen, Germany.;Counago, RM (通讯作者),Univ Estadual Campinas, Ctr Biol Mol & Engn Genet CBMEG, Ctr Quim Med CQMED, UNICAMP, BR-13083875 Campinas, SP, Brazil.;Counago, RM (通讯作者),Univ Estadual Campinas, Inst Biol, Dept Genet & Evolucao, Struct Genom Consortium, BR-13083886 Campinas, SP, Brazil.;Gehringer, M (通讯作者),Univ Tubingen, Cluster Excellence iFIT EXC 2180 Image Guided & F, D-72076 Tubingen, Germany.
JOURNAL OF MEDICINAL CHEMISTRY, 2022; 65 (4): 3173