Design, synthesis, and biological evaluation of pyrrolopyrimidine derivatives as novel Bruton?s tyrosine kinase (BTK) inhibitors

Yang, MJ; Jiang, HM; Yang, Z; Liu, X; Sun, HY; Hao, MY; Hu, JP; Chen, XG; Jin, J; Wang, XJ

Chen, XG; Jin, J; Wang, XJ (通讯作者),Peking Union Med Coll & Chinese Acad Med Sci, Inst Mat Med, State Key Lab Bioact Subst & Funct Nat Med, Beijing 100050, Peoples R China.;Hu, JP (通讯作者),Chinese Acad Med Sci & Peking Union Med Coll, Beijing Key Lab Nonclin Drug Metab & PK, PD Study, Beijing 100050, Peoples R China.

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022; 241 ():

Abstract

Developing Bruton's tyrosine kinase (BTK) inhibitors has become a significant focus in recent years because BTK inhibition is an effective approach fo......

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