Highly enantioselective enantioselective Biginelli reactions using methanopyroline/thiourea - based dual organocatalyst systems: asymmetric synthesis of 4-substituted unsaturated aryl dihydropyrimidines

Yu, H; Xu, P; He, HH; Zhu, J; Lin, HL; Han, S

Yu, H; Han, S (reprint author), Shanghai Inst Technol, Sch Chem & Environm Engn, Shanghai 201418, Peoples R China.; Yu, H (reprint author), Tsinghua Univ, Dept Chem, Beijing 100084, Peoples R China.

TETRAHEDRON-ASYMMETRY, 2017; 28 (2): 257

Abstract

A series of novel chiral 3,4-dihydropyrimidin-2-(1H)-ones and -thiones (DHPMs) was developed via asymmetric Biginelli reactions catalyzed by a methano......

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