Bidirectional modulation of HIF-2 activity through chemical ligands

Wu, DL; Su, XY; Lu, JP; Li, S; Hood, BL; Vasile, S; Potluri, N; Diao, XT; Kim, Y; Khorasanizadeh, S; Rastinejad, F

Wu, DL (reprint author), Shandong Univ, Helmholtz Int Lab, State Key Lab Microbial Technol, Qingdao, Peoples R China.; Wu, DL; Rastinejad, F (reprint author), Sanford Burnham Prebys Med Discovery Inst, Integrat Metab Program, Orlando, FL 92037 USA.; Rasti

NATURE CHEMICAL BIOLOGY, 2019; 15 (4): 367

Abstract

Hypoxia-inducible factor-2 (HIF-2) is a heterodimeric transcription factor formed through dimerization between an oxygen-sensitive HIF-2 alpha subunit......

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