Determination and pharmacokinetic study of AZD-3759 in rat plasma by ultra performance liquid chromatography with triple quadrupole mass spectrometer

Wu, QJ; Hua, AL; Sun, YG; Ma, C; Tian, WX; Huang, C; Yu, HB; Jiao, P; Wang, SH; Tong, HF; Qiu, WW

Tong, HF (reprint author), Beijing Hosp, Dept Thorac Surg, Natl Ctr Gerontol, 1 Dahua Rd, Beijing 100730, Peoples R China.; Qiu, WW (reprint author), Wenzhou Med Univ, Peoples Hosp Lishui, Affiliated Hosp 6, Dept Neurol, 15 Dazhong St, Lishui 323000, Peop

THORACIC CANCER, 2018; 9 (11): 1383

Abstract

Background Methods AZD-3759 is a new, potent, oral, active central nervous system-penetrant EGFR inhibitor. Despite promising clinical activity among ......

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