K2S2O8-Activated Friedel-Crafts Type Alkylation of Indoles with alpha-Amido Sulfones

Wu, XY; Xue, L; Luo, SL; Jia, SQ; Ao, J; Qin, WL

Qin, WL (reprint author), Chongqing Univ, Sch Pharmaceut Sci, Innovat Drug Res Ctr, 55 Daxuecheng,South Rd, Chongqing 401331, Peoples R China.

SYNTHESIS-STUTTGART, 2017; 49 (22): 5017

Abstract

A K2S2O8-activated regioselective alkylation of alpha-amido sulfones at the C-3 position of indoles is reported. The protocol developed herein provide......

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