A novel RRGW derived peptide is a promising inhibitor of BoNT/A

Ma, WT; Wang, LL; Tan, XM; Wang, X; Yang, CY; Wang, Y; Liu, ZY; Liu, B; Zhu, H; Zhi, DJ; Wang, DS

Zhi, DJ; Wang, DS (通讯作者),Lanzhou Univ, Sch Pharm, 199 West Donggang Rd, Lanzhou 730000, Peoples R China.

JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 2023; 38 (1):

Abstract

Clostridium botulinum neurotoxin type A (BoNT/A) is one of the most potent biotoxins ever known. Its entry into neurons could block vesicle exocytosis......

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