Open channel block of Kv1.5 channels by HMQ1611

Dong, C; Li, JW; Ding, WG; Ueda, R; Xie, XL; Wu, J; Matsuura, H; Horie, M

Wu, J (通讯作者),Xian Jiaotong Univ Hlth Sci Ctr, Sch Basic Med Sci, Dept Pharmacol, Xian, Shaanxi, Peoples R China.;Wu, J (通讯作者),Xi An Jiao Tong Univ, Key Lab Environm & Genes Related Dis, Minist Educ, Xian, Shaanxi, Peoples R China.;Wu, J (通讯作者),Shiga Univ Med Sci, Dept Physiol, Otsu, Shiga, Japan.;Wu, J (通讯作者),Shiga Univ Med Sci, Dept Cardiovasc & Resp Med, Otsu, Shiga, Japan.

FRONTIERS IN PHARMACOLOGY, 2022; 13 ():

Abstract

Kv1.5 channels conduct the ultra-rapid delayed rectifier potassium current (I (Kur)). Pharmacological blockade of human Kv1.5 (hKv1.5) has been regard......

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