Optimization of antimalarial, and anticancer activities of (E)-methyl 2-(7-chloroquinolin-4-ylthio)-3-(4-hydroxyphenyl) acrylate

Romero, JA; Acosta, ME; Gamboa, ND; Mijares, MR; De Sanctis, JB; Charris, JE

Charris, JE (reprint author), Univ Cent Venezuela, Fac Farm, Unidad Bioquim, Lab Sintesis Organ, Apartado 47206, Caracas 1041A, Venezuela.

BIOORGANIC & MEDICINAL CHEMISTRY, 2018; 26 (4): 815

Abstract

Chemically modified versions of bioactive substances, are particularly useful in overcoming barriers associated with drug formulation, drug delivery a......

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