Tuned out

Ferguson, FM

Ferguson, FM (通讯作者),Univ Calif San Diego, Dept Chem & Biochem, San Diego, CA 92103 USA.;Ferguson, FM (通讯作者),Univ Calif San Diego, Skaggs Sch Pharm & Pharmaceut Sci, San Diego, CA 92103 USA.

NATURE CHEMICAL BIOLOGY, 2022; 18 (9): 917

Abstract

Controlling kinase inhibitors' residence time via reversible covalent binding is of high interest in drug discovery. Tuning reversible covalent bindin......

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