Dihydropyridine Lactam Analogs Targeting BET Bromodomains

Jiang, JW; Sigua, LH; Chan, A; Kalra, P; Pomerantz, WCK; Schonbrunn, E; Qi, J; Georg, GI

Georg, GI (通讯作者)，Univ Minnesota, Coll Pharm, Dept Med Chem, 717 Delaware St SE, Minneapolis, MN 55414 USA.;Georg, GI (通讯作者)，Univ Minnesota, Coll Pharm, Inst Therapeut Discovery & Dev, 717 Delaware St SE, Minneapolis, MN 55414 USA.

CHEMMEDCHEM, 2022; 17 (1):

Abstract

Inhibitors of Bromodomain and Extra Terminal (BET) proteins are investigated for various therapeutic indications, but selectivity for BRD2, BRD3, BRD4......

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