Palladium-Catalyzed Regioselective C-H Arylation of 4-Azaindazole at C3, C5 and C7 Positions

Faarasse, S; El Kazzouli, S; Bourzikat, O; Bourg, S; Aci-Seche, S; Bonnet, P; Suzenet, F; Guillaumet, G

Suzenet, F; Guillaumet, G (corresponding author), Univ Orleans, Inst Organ & Analyt Chem, CNRS, UMR 7311, BP 6759, F-45067 Orleans 2, France.; El Kazzouli, S; Guillaumet, G (corresponding author), Euromed Univ Fes UEMF, Sch Engn Biomed & Biotechnol, Euromed Res Ctr, Route Meknes, Fes 30000, Morocco.

ADVANCED SYNTHESIS & CATALYSIS, ; ():

Abstract

Direct and site-selective C5 and C7 palladium-catalyzed C-H arylations of 4-azaindazole N-oxide have been achieved. A bidentate ligand and Pd(OAc)(2) ......

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