Quadruple Target Evaluation of Diversity-Optimized Halogen-Enriched Fragments (HEFLibs) Reveals Substantial Ligand Efficiency for AP2-Associated Protein Kinase 1 (AAK1)

Dammann, M; Kramer, M; Zimmermann, MO; Boeckler, FM

Boeckler, FM (通讯作者),Eberhard Karls Univ Tubingen, Inst Pharmaceut Sci, Dept Biochem & Pharm, Lab Mol Design & Pharmaceut Biophys, Tubingen, Germany.;Boeckler, FM (通讯作者),Eberhard Karls Univ Tubingen, Interfac Inst Biomed Informat IBMI, Tubingen, Germany.

FRONTIERS IN CHEMISTRY, 2022; 9 ():