Non-small molecule PROTACs (NSM-PROTACs): Protein degradation kaleidoscope

Ma, SN; Ji, JA; Tong, YY; Zhu, YX; Dou, JW; Zhang, X; Xu, SC; Zhu, TB; Xu, XL; You, QD; Jiang, ZY

Xu, XL; You, QD; Jiang, ZY (通讯作者),China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China.;Xu, XL; You, QD; Jiang, ZY (通讯作者),China Pharmaceut Univ, Jiang Su Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China.;Xu, XL; You, QD; Jiang, ZY (通讯作者),China Pharmaceut Univ, Sch Pharm, Dept Med Chem, Nanjing 210009, Peoples R China.

ACTA PHARMACEUTICA SINICA B, 2022; 12 (7): 2990

Abstract

The proteolysis targeting chimeras (PROTACs) technology has been rapidly developed since its birth in 2001, attracting rapidly growing attention of sc......

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