Phthalimide-tethered isatins as novel poly(ADP-ribose) polymerase inhibitors: Design, synthesis, biological evaluations, and molecular modeling investigations

El Hassab, MA; El-Hafeez, AAA; Almahli, H; Elsayed, ZM; Eldehna, WM; Hassan, GS; Abou-Seri, SM

El-Hafeez, AAA (通讯作者),Cairo Univ, Natl Canc Inst, Canc Biol Dept, Pharmacol & Expt Oncol Unit, Cairo, Egypt.;Eldehna, WM (通讯作者),Kafrelsheikh Univ, Fac Pharm, Dept Pharmaceut Chem, Kafrelsheikh 33516, Egypt.;Abou-Seri, SM (通讯作者),Cairo Univ, Fac Pharm, Pharmaceut Chem Dept, Cairo 11562, Egypt.

ARCHIV DER PHARMAZIE, 2023; ():

Abstract

Humanity is currently facing various diseases with significant mortality rates, particularly those associated with malignancies. Numerous enzymes and ......

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