Design, synthesis and biological evaluation of dipeptides as novel non-covalent 20S proteasome inhibitors

Yang, YJ; Wang, K; Yang, Y; Lai, FF; Chen, XG; Xiao, ZY

Xiao, ZY (corresponding author), Chinese Acad Med Sci & Peking Union Med Coll, Inst Mat Med, Beijing Key Lab Active Subst Discovery & Druggabi, Beijing 100050, Peoples R China.

JOURNAL OF ASIAN NATURAL PRODUCTS RESEARCH, 2021; 23 (5): 436

Abstract

Based on the interaction modes of the natural 20S proteasome inhibitors TMC-95A, we have previously discovered a dipeptide 1. To explore the SAR aroun......

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