Neratinib is a TFEB and TFE3 activator that potentiates autophagy and unbalances energy metabolism in ERBB2+breast cancer cells

Bellese, G; Tagliatti, E; Gagliani, MC; Santamaria, S; Arnaldi, P; Falletta, P; Rusmini, P; Matteoli, M; Castagnola, P; Cortese, K

Cortese, K (通讯作者),Univ Genoa, Dept Expt Med, Cellular Electron Microscopy Lab, DIMES, Genoa, Italy.;Castagnola, P (通讯作者),IRCCS Osped Policlin San Martino, Genoa, Italy.

BIOCHEMICAL PHARMACOLOGY, 2023; 213 ():

Abstract

Neratinib (NE) is an irreversible pan-ERBB tyrosine kinase inhibitor used to treat breast cancers (BCa) with amplification of the ERBB2/HER2/Neu gene ......

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