Identification of ritanserin analogs that display DGK isoform specificity

Granade, ME; Manigat, LC; Lemke, MC; Purow, BW; Harris, TE

Harris, TE (通讯作者),Univ Virginia, Sch Med, Dept Pharmacol, Charlottesville, VA 22908 USA.;Purow, BW (通讯作者),Univ Virginia, Dept Neurol, Div Neurooncol, Charlottesville, VA 22904 USA.

BIOCHEMICAL PHARMACOLOGY, 2022; 197 ():

Abstract

The diacylglycerol kinase (DGK) family of lipid enzymes catalyzes the conversion of diacylglycerol (DAG) to phosphatidic acid (PA). Both DAG and PA ar......

Full Text Link