Discovery and in vitro characterization of AMG 510-a potent and selective covalent small-molecule inhibitor of KRAS(G12C)

Saiki, AY; Gaida, K; Rex, K; Achanta, P; San Miguel, T; Koppada, N; Bagal, D; Lanman, BA; Foti, RS; McCarter, JD; Volak, LP; Canon, J; Cee, VJ; Lipford, JR

CANCER RESEARCH, 2019; 79 (13):