Identification of Slow-Binding Inhibitors of the BoNT/A Protease

Patel, EN; Turner, LD; Hixon, MS; Janda, KD

Janda, KD (通讯作者),Scripps Res Inst, Skaggs Inst Chem Biol, Worm Inst Res & Med WIRM, Dept Chem, La Jolla, CA 92037 USA.;Janda, KD (通讯作者),Scripps Res Inst, Skaggs Inst Chem Biol, Worm Inst Res & Med WIRM, Dept Immunol, La Jolla, CA 92037 USA.

ACS MEDICINAL CHEMISTRY LETTERS, 2022; 13 (4): 742

Abstract

Botulinum neurotoxin A (BoNT/A) is a lethal toxin, which causesbotulism, and is categorized as a bioterrorism threat, which causesflaccid paralysisand......

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