An Activator-Blocker Pair Provides a Controllable On-Off Switch for a Ketosteroid Isomerase Active Site Mutant

Lamba, V; Yabukarski, F; Herschlag, D

Herschlag, D (reprint author), Stanford Univ, Dept Biochem, Stanford, CA 94305 USA.; Herschlag, D (reprint author), Stanford Univ, Dept Chem, Stanford, CA 94305 USA.; Herschlag, D (reprint author), Stanford Univ, Dept Chem Engn, Stanford, CA 94305 USA.; H

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2017; 139 (32): 11089

Abstract

Control of enzyme activity is fundamental to biology and represents a long-term goal in bioengineering and precision therapeutics. While several power......

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