Pharmacokinetic and Pharmacodynamic Studies of Elacestrant, A Novel Oral Selective Estrogen Receptor Degrader, in Healthy Post-Menopausal Women

Conlan, MG; de Vries, EFJ; Glaudemans, AWJM; Wang, YM; Troy, S

Conlan, MG (corresponding author), Radius Hlth Inc, Dept Oncol Clin Dev, 950 Winter St, Waltham, MA 02451 USA.

EUROPEAN JOURNAL OF DRUG METABOLISM AND PHARMACOKINETICS, 2020; 45 (5): 675

Abstract

Background and Objectives Advanced estrogen receptor-positive (ER+) breast cancer is currently treated with endocrine therapy. Elacestrant is a novel,......

Full Text Link