Discovery of Rogaratinib (BAY 1163877): a pan-FGFR Inhibitor

Collin, MP; Lobell, M; Hubsch, W; Brohm, D; Schirok, H; Jautelat, R; Lustig, K; Bomer, U; Vohringer, V; Heroult, M; Grunewald, S; Hess-Stumpp, H

Collin, MP (reprint author), Bayer AG, Drug Discovery, Dept Med Chem, Postfach 101709, D-42096 Wuppertal, Germany.

CHEMMEDCHEM, 2018; 13 (5): 437

Abstract

Rogaratinib (BAY 1163877) is a highly potent and selective small-molecule pan-fibroblast growth factor receptor (FGFR) inhibitor (FGFR1-4) for oral ap......

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