A Comparison of the Pharmacokinetics and Safety of Dapagliflozin Formate, an Ester Prodrug of Dapagliflozin, to Dapagliflozin Propanediol Monohydrate in Healthy Subjects

Kim, HC; Lee, S; Sung, S; Kim, E; Jang, IJ; Chung, JY

Chung, JY (通讯作者),Seoul Natl Univ, Coll Med, Seongnam Si 13620, Gyeonggi Do, South Korea.;Chung, JY (通讯作者),Bundang Hosp, Seongnam Si 13620, Gyeonggi Do, South Korea.

DRUG DESIGN DEVELOPMENT AND THERAPY, 2023; 17 (): 1203

Abstract

Background: Dapagliflozin formate (DAP-FOR, DA-2811), an ester prodrug of dapagliflozin, was developed to improve the stability and pharmaceutical man......

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