Enterovirus inhibitory activity of C-8-tert-butyl substituted 4-aryl-6,7,8,9-tetrahydrobenzo[4,5]thieno[3,2-e][1,2,4]triazolo[4,3-a]pyrimidin-5(4H)-ones

Biswas, BK; Malpani, YR; Ha, N; Kwon, DH; Shin, JS; Kim, HS; Kim, C; Han, SB; Lee, CK; Jung, YS

Jung, YS (reprint author), Korea Res Inst Chem Technol, Bio & Drug Discovery Div, 141 Gajeongro, Yuseong 34114, Daejeon, South Korea.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2017; 27 (15): 3582

Abstract

Members of a series of 4-aryl-6,7,8,9-tetrahydrobenzo[ 4,5] thieno[ 3,2-e][ 1,2,4] triazolo[ 4,3-a] pyrimidin-5 (4H)-ones (1, Fig. 2) were prepared an......

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