Novel 6-aryl substituted 4-pyrrolidineaminoquinazoline derivatives as potent phosphoinositide 3-kinase delta (PI3K delta) inhibitors

Xin, MH; Duan, WM; Feng, YF; Hei, YY; Zhang, H; Shen, Y; Zhao, HY; Mao, S; Zhang, SQ

Zhang, SQ (reprint author), Xi An Jiao Tong Univ, Hlth Sci Ctr, Sch Pharm, Dept Med Chem, 76 West Yanta Rd, Xian 710061, Shaanxi, Peoples R China.

BIOORGANIC & MEDICINAL CHEMISTRY, 2018; 26 (8): 2028

Abstract

In this study, a novel series of 6-aryl substituted 4-pyrrolidineaminoquinazoline derivatives were designed and evaluated as potent PI3K delta inhibit......

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