Thiophene bioisosteres of GluN2B selective NMDA receptor antagonists: Synthesis and pharmacological evaluation of [7]annuleno[b]thiophen-6-amines

Baumeister, S; Schepmann, D; Wunsch, B

Wunsch, B (corresponding author), Westfalische Wilhelms Univ Munster, Inst Pharmazeut & Med Chem, Corrensstr 48, D-48149 Munster, Germany.

BIOORGANIC & MEDICINAL CHEMISTRY, 2020; 28 (2):

Abstract

Thiophene bioisosteres of potent GluN2B receptor negative allosteric modulators were prepared and evaluated pharmacologically. The five-step synthesis......

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