LSD1 inhibitors for cancer treatment: Focus on multi-target agents and compounds in clinical trials

Noce, B; Di Bello, E; Fioravanti, R; Mai, A

Fioravanti, R (通讯作者),Sapienza Univ Rome, Dept Chem & Technol Drugs, Rome, Italy.

FRONTIERS IN PHARMACOLOGY, 2023; 14 ():

Abstract

Histone lysine-specific demethylase 1 (LSD1/KDM1A) was first identified in 2004 as an epigenetic enzyme able to demethylate specific lysine residues o......

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