Identification of a Protein Arginine Methyltransferase 7 (PRMT7)/Protein Arginine Methyltransferase 9 (PRMT9) Inhibitor

Feoli, A; Iannelli, G; Cipriano, A; Milite, C; Shen, L; Wang, ZH; Hadjikyriacou, A; Lowe, TL; Safaeipour, C; Viviano, M; Sarno, G; Morretta, E; Monti, MC; Yang, YZ; Clarke, SG; Cosconati, S; Castellano, S; Sbardella, G

Castellano, S; Sbardella, G (通讯作者),Univ Salerno, Dept Pharm, Epigenet Med Chem Lab, I-84084 Fisciano, SA, Italy.;Cosconati, S (通讯作者),Univ Campania Luigi Vanvitelli, DiSTABiF, I-81100 Caserta, Italy.

JOURNAL OF MEDICINAL CHEMISTRY, 2023; 66 (19): 13665

Abstract

Less studied than the other protein arginine methyltransferaseisoforms, PRMT7 and PRMT9 have recently been identified as importanttherapeutic targets.......

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