Strategies to overcome resistance mutations of Bruton's tyrosine kinase inhibitor ibrutinib

Liu, LY; Shi, BY; Wang, XQ; Xiang, H

Xiang, H (reprint author), China Pharmaceut Univ, Jiangsu Key Lab Drug Design & Optimizat, 24 Tongjiaxiang, Nanjing 210009, Jiangsu, Peoples R China.; Xiang, H (reprint author), China Pharmaceut Univ, Sch Pharm, Dept Med Chem, 24 Tongjiaxiang, Nanjing 210

FUTURE MEDICINAL CHEMISTRY, 2018; 10 (3): 343

Abstract

Ibrutinib, as the first Bruton's tyrosine kinase (Btk) inhibitor, has been shown to have clinically significant activity in leukemias and lymphomas. H......

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