Chemoprobe-based assays of histone lysine demethylase 1A target occupation enable in vivo pharmacokinetics and pharmacodynamics studies of KDM1A inhibitors

Mascaro, C; Ortega, A; Carceller, E; Rodriguez, RR; Ciceri, F; Lunardi, S; Yu, L; Hilbert, M; Maes, T

Maes, T (reprint author), Oryzon Genom SA, Carrer St Ferran 74, Barcelona 08940, Spain.

JOURNAL OF BIOLOGICAL CHEMISTRY, 2019; 294 (20): 8311