Crystallization-Based Synthetic Route to Antimalarial Agent BRD5018: Diazocene Ring Formation via a Staudinger-aza-Wittig Reaction on an Azetidine-Ribose Template

Mitasev, B; Yang, J; Gusovsky, F; Girish, D; Khile, AS; Balla, VS; Vikram, V; Vaddi, A; Bathula, S; Sugandham, SR; Terli, C; Kalla, V; Rayaprolu, PK; Talabhakthula, RK; Gotoda, M; Melillo, B; Schreiber, SL; Fang, FG

Mitasev, B; Fang, FG (通讯作者),G2D2 Eisai Inc, Cambridge, MA 02140 USA.

ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2022; 26 (3): 817