Effective Activation of BKCa Channels by QO-40 (5-(Chloromethyl)-3-(Naphthalen-1-yl)-2-(Trifluoromethyl)Pyrazolo [1,5-a]pyrimidin-7(4H)-one), Known to Be an Opener of KCNQ2/Q3 Channels

Chang, WT; Wu, SN

Wu, SN (corresponding author), Natl Cheng Kung Univ, Med Coll, Dept Physiol, Tainan 70101, Taiwan.; Wu, SN (corresponding author), Natl Cheng Kung Univ, Med Coll, Inst Basic Med Sci, Tainan 70101, Taiwan.; Wu, SN (corresponding author), China Med Univ, China Med Univ Hosp, Dept Med Res, Taichung 40402, Taiwan.

PHARMACEUTICALS, 2021; 14 (5):

Abstract

QO-40 (5-(chloromethyl)-3-(naphthalene-1-yl)-2-(trifluoromethyl) pyrazolo[1,5-a]pyrimidin-7(4H)-one) is a novel and selective activator of KCNQ2/KCNQ3......

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