Discovery of Novel Gq-Biased LPA1 Negative Allosteric Modulators

Shimizu, Y; Nakayama, M

Shimizu, Y (reprint author), Takeda Pharmaceut Co Ltd, Pharmaceut Res Div, Biomol Res Labs, 26-1 Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, Japan.

SLAS DISCOVERY, 2017; 22 (7): 859

Abstract

Lysophosphatidic acid (LPA) activates the G-protein-coupled receptor LPA1, which regulates various cellular processes, including cell proliferation an......

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