The D647N mutation of FGFR1 induces ligand-independent receptor activation

Domenichini, M; Ravelli, C; Corsini, M; Codenotti, S; Moreschi, E; Gogna, A; Capoferri, D; Zizioli, D; Bresciani, R; Grillo, E; Mitola, S

Grillo, E; Mitola, S (通讯作者),Univ Brescia, Dept Mol & Translat Med, Viale Europa 11, I-25123 Brescia, Italy.

BIOCHIMICA ET BIOPHYSICA ACTA-GENERAL SUBJECTS, 2023; 1867 (12):

Abstract

The activation loop (A-loop) of kinases, a key regulatory region, is recurrently mutated in several kinase proteins in cancer resulting in dysregulate......

Full Text Link