Physiologically Based Pharmacokinetic Modeling of Palbociclib

Yu, YK; Loi, CM; Hoffman, J; Wang, DN

Yu, YK (reprint author), Pfizer La Jolla, Clin Pharmacol, Global Prod Dev, 10555 Sci Ctr Dr, San Diego, CA 92121 USA.

JOURNAL OF CLINICAL PHARMACOLOGY, 2017; 57 (2): 173

Abstract

Palbociclib is an orally available CDK4/6 inhibitor. In humans, palbociclib undergoes metabolism mediated primarily by CYP3A and SULT2A1, and it is al......

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