Synthesis and biological screening of new thiazolo[4,5-d] pyrimidine and dithiazolo[3,2-a:5 ',4 '-e]pyrimidinone derivatives as antimicrobial, antiquorum-sensing and antitumor agents

Abd Elhameed, AA; El-Gohary, NS; El-Bendary, ER; Shaaban, MI; Bayomi, SM

El-Gohary, NS (reprint author), Mansoura Univ, Fac Pharm, Dept Med Chem, Mansoura 35516, Egypt.

BIOORGANIC CHEMISTRY, 2018; 81 (): 299

Abstract

New thiazolopyrimidine and dithiazolopyrimidinone derivatives 2-11 were synthesized and estimated for antimicrobial activity against S. aureus, B. cer......

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